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La chinasi 5 del recettore accoppiato alla proteina G media la soppressione della crescita indotta dal gene 1 indotta dal tazarotene delle cellule di cancro del colon umano.La chinasi 5 del recettore accoppiato alla proteina G media la soppressione della crescita indotta dal gene 1 indotta dal tazarotene delle cellule di cancro del colon umano.

La chinasi 5 del recettore accoppiato alla proteina G media la soppressione della crescita indotta dal gene 1 indotta dal tazarotene delle cellule di cancro del colon umano.

Posted on Dicembre 4, 2020 By andrea Nessun commento su La chinasi 5 del recettore accoppiato alla proteina G media la soppressione della crescita indotta dal gene 1 indotta dal tazarotene delle cellule di cancro del colon umano.

SFONDO
Il gene 1 indotto da tazarotene (TIG1) è un gene soppressore tumorale di tipo II inducibile dai retinoidi. L’isoforma B di TIG1 (TIG1B) inibisce la crescita e l’invasione delle cellule tumorali. L’espressione di TIG1B è spesso sottoregolata in vari tessuti tumorali; tuttavia, l’espressione e le attività dell’isoforma TIG1A devono ancora essere riportate. Pertanto, questo studio ha esaminato gli effetti delle isoforme TIG1A e TIG1B sulla crescita cellulare e sui profili di espressione genica utilizzando cellule di cancro del colon.

METODI
I cloni stabili TIG1A e TIG1B derivati ​​da cellule di cancro al colon HCT116 e SW620 sono stati stabiliti utilizzando il sistema GeneSwitch; L’espressione dell’isoforma TIG1 è stata indotta dal trattamento con mifepristone. La crescita cellulare è stata valutata utilizzando i test di proliferazione cellulare e formazione di colonie WST-1. L’interferenza dell’RNA è stata utilizzata per esaminare i cambiamenti di mediazione di TIG1 nella crescita cellulare. I profili di espressione genica sono stati determinati utilizzando microarray e convalidati utilizzando la reazione a catena della polimerasi in tempo reale e analisi Western blot.

RISULTATI
Entrambe le isoforme di TIG1 sono state espresse a livelli elevati nei tessuti normali della prostata e del colon e sono state sottoregolate nelle linee cellulari di cancro del colon. Entrambe le isoforme TIG1 hanno inibito in modo significativo la crescita di cellule HCT116 transitoriamente trasfettate ed esprimendo stabilmente cellule TIG1A e TIG1B HCT116 e SW620. L’espressione dei geni 129 e 55 è stata alterata all’induzione dell’espressione di TIG1A e TIG1B, rispettivamente, nelle cellule HCT116 che esprimono stabilmente. Dei geni analizzati, 23 e 6 geni erano rispettivamente sovraregolati e sottoregolati nelle cellule che esprimono TIG1A e TIG1B. La sovraregolazione della chinasi 5 del recettore accoppiato alla proteina G (GRK5) è stata confermata utilizzando la reazione a catena della polimerasi in tempo reale e analisi Western blot in entrambe le linee cellulari stabili TIG1. Il silenziamento dell’espressione di TIG1A o GRK5 ha ridotto significativamente la soppressione della crescita cellulare mediata da TIG1A.

CONCLUSIONI
L’espressione di entrambe le isoforme di TIG1 è stata osservata nei tessuti normali della prostata e del colon ed è stata sottoregolata nelle linee cellulari di cancro del colon. Entrambe le isoforme TIG1 hanno soppresso la crescita cellulare e stimolato l’espressione di GRK5 nelle cellule HCT116 e SW620. Il knockdown dell’espressione di GRK5 ha alleviato la soppressione della crescita indotta da TIG1A delle cellule HCT116, suggerendo che GRK5 media la soppressione della crescita cellulare da parte di TIG1A. Pertanto, TIG1 può partecipare alla sottoregolazione della segnalazione accoppiata alla proteina G sovraregolando l’espressione di GRK5.

 

Metodi spettrofotometrici che indicano la stabilità per la determinazione del tazarotene in presenza del suo prodotto di degradazione alcalino mediante tecniche spettrofotometriche derivate.

È stata studiata la stabilità del tazarotene (TZ) e sono stati utilizzati due metodi di indicazione della stabilità, vale a dire, il derivato primo e un metodo spettrofotometrico del rapporto dei derivati, per determinare il tazarotene in presenza del suo prodotto di degradazione alcalina (HD) utilizzando metanolo come solvente. È stata ottenuta una relazione lineare nell’intervallo 1-10 µg ml ¹ per entrambi i metodi.

Applicando i metodi proposti, è stato possibile determinare il tazarotene nella sua polvere pura da con precisione 99,35 ± 1,410 (n = 10) per il metodo della derivata prima e 99,45 ± 1,053 (n = 10) per il metodo del rapporto dei derivati. I metodi del derivato primo e del rapporto dei derivati ​​sono stati utilizzati per l’analisi di miscele preparate in laboratorio contenenti diversi rapporti di tazarotene e del suo prodotto di degradazione ed erano validi in presenza rispettivamente fino al 70% e all’80% di prodotto di degradazione. I metodi proposti sono stati convalidati e trovati adatti come metodi di analisi indicanti la stabilità per il tazarotene in formulazioni farmaceutiche.

La chinasi 5 del recettore accoppiato alla proteina G media la soppressione della crescita indotta dal gene 1 indotta dal tazarotene delle cellule di cancro del colon umano.La chinasi 5 del recettore accoppiato alla proteina G media la soppressione della crescita indotta dal gene 1 indotta dal tazarotene delle cellule di cancro del colon umano.
La chinasi 5 del recettore accoppiato alla proteina G media la soppressione della crescita indotta dal gene 1 indotta dal tazarotene delle cellule di cancro del colon umano.

[Retinoidi: meccanismi d’azione].

I retinoidi, derivati ​​della vitamina A, sono molecole naturali o sintetiche con effetti pleiotropici, che regolano il differenziamento, la proliferazione e l’apoptosi cellulare. Nella cellula bersaglio, i metaboliti naturali attivi acido retinoico (RA) e acido 9-cis-retinoico sono sintetizzati dal retinolo mediante un processo in due fasi con il metabolita intermedio retinaldeide. Nel 1987, l’identificazione dei recettori nucleari dell’acido retinoico che appartengono alla superfamiglia dei recettori nucleari ha portato a un progresso significativo nella comprensione del meccanismo d’azione dei retinoidi. Esistono due famiglie di recettori nucleari retinoidi (RNR), i recettori RA (RAR), il cui ligando naturale è RA, e i recettori X retinoidi (RXR), il cui ligando naturale è acido 9-cis-retinoico. Tra i retinoidi sintetici, isotretinoina, acitretina, tazarotene e adapalene sono ligandi del RAR, il bexarotene è il primo rexinoide (ligando dell’RXR), l’alitretinoina il primo panagonista (RAR + RXR).

Tissue Factor Recombinant Rabbit mAb

BS48470 Bioworld Biotech 50 ul 398 EUR
Description: Store at -20°C. Supplied in 50mM Tris-Glycine(pH 7.4), 0.15M NaCl, 40%Glycerol, 0.01% sodium azide and 0.05% BSA. Stable for 12 months from date of receipt.

Tissue Factor Recombinant Rabbit mAb

BS46451 Bioworld Biotech 50 ul 398 EUR
Description: Store at -20°C. Supplied in 50mM Tris-Glycine(pH 7.4), 0.15M NaCl, 40%Glycerol, 0.01% sodium azide and 0.05% BSA. Stable for 12 months from date of receipt.

Tissue Factor Recombinant Rabbit mAb

BS45077 Bioworld Biotech 50 ul 398 EUR
Description: Store at -20°C. Supplied in 50mM Tris-Glycine(pH 7.4), 0.15M NaCl, 40%Glycerol, 0.01% sodium azide and 0.05% BSA. Stable for 12 months from date of receipt.

Tissue Factor Recombinant Rabbit mAb

BS45170 Bioworld Biotech 50 ul 398 EUR
Description: Store at -20°C. Supplied in 50mM Tris-Glycine(pH 7.4), 0.15M NaCl, 40%Glycerol, 0.01% sodium azide and 0.05% BSA. Stable for 12 months from date of receipt.

Tissue factor Recombinant Rabbit mAb

E47M52647 EnoGene 100ul 495 EUR

Recombinant Rabbit Tissue factor (F3), partial

MBS7111604-INQUIRE MyBiosource INQUIRE Ask for price

Recombinant Rabbit Tissue factor pathway inhibitor

MBS9422521-002mg MyBiosource 0.02mg 505 EUR

Recombinant Rabbit Tissue factor pathway inhibitor

MBS9422521-01mg MyBiosource 0.1mg 895 EUR

Recombinant Rabbit Tissue factor pathway inhibitor

MBS9422521-05mg MyBiosource 0.5mg 1975 EUR

Recombinant Rabbit Tissue factor pathway inhibitor

MBS9422521-5x05mg MyBiosource 5x0.5mg 8735 EUR

Recombinant Rabbit Tissue factor pathway inhibitor

MBS9420734-002mg MyBiosource 0.02mg 460 EUR

Recombinant Rabbit Tissue factor pathway inhibitor

MBS9420734-01mg MyBiosource 0.1mg 795 EUR

Recombinant Rabbit Tissue factor pathway inhibitor

MBS9420734-1mg MyBiosource 1mg 2525 EUR

Recombinant Rabbit Tissue factor pathway inhibitor

MBS9420734-5x1mg MyBiosource 5x1mg 11205 EUR

Recombinant Rabbit Tissue factor pathway inhibitor (TFPI)

CSB-EP023437RB Cusabio 2318 mg Ask for price

Recombinant Rabbit Tissue factor pathway inhibitor (TFPI)

CSB-EP023437RB-20ug Cusabio 20ug Ask for price
Description: 25-300aa

Recombinant Rabbit Tissue factor pathway inhibitor(TFPI)

AP70839 SAB 1mg 2826 EUR

Recombinant Rabbit Tissue factor pathway inhibitor(TFPI)

AP72812 SAB each Ask for price

Recombinant Rabbit Tissue factor pathway inhibitor (TFPI)

CSB-BP023437RB Cusabio 118 mg Ask for price

Recombinant Rabbit Tissue factor pathway inhibitor (TFPI)

CSB-BP023437RB-20ug Cusabio 20ug Ask for price
Description: 25-300aa

Recombinant Rabbit Tissue factor pathway inhibitor (TFPI)

CSB-YP023437RB Cusabio 6035 mg Ask for price

Recombinant Rabbit Tissue factor pathway inhibitor (TFPI)

CSB-YP023437RB-20ug Cusabio 20ug Ask for price
Description: 25-300aa

Recombinant Rabbit Tissue factor pathway inhibitor (TFPI)

MBS956430-002mgBaculovirus MyBiosource 0.02mg(Baculovirus) 475 EUR

Recombinant Rabbit Tissue factor pathway inhibitor (TFPI)

MBS956430-002mgEColi MyBiosource 0.02mg(E-Coli) 375 EUR

Recombinant Rabbit Tissue factor pathway inhibitor (TFPI)

MBS956430-002mgMammalianCell MyBiosource 0.02mg(Mammalian-Cell) 580 EUR

Recombinant Rabbit Tissue factor pathway inhibitor (TFPI)

MBS956430-002mgYeast MyBiosource 0.02mg(Yeast) 420 EUR

Recombinant Rabbit Tissue factor pathway inhibitor (TFPI)

MBS956430-01mgEColi MyBiosource 0.1mg(E-Coli) 635 EUR

Recombinant Rabbit Tissue factor pathway inhibitor (TFPI)

RPC22103-100ug Biomatik Corporation 100ug 721.6 EUR

Recombinant Rabbit Tissue factor pathway inhibitor (TFPI)

RPC22103-1mg Biomatik Corporation 1mg 2884.7 EUR

Recombinant Rabbit Tissue factor pathway inhibitor (TFPI)

RPC22103-20ug Biomatik Corporation 20ug 448.1 EUR

Recombinant Rabbit Tissue factor pathway inhibitor (TFPI)

RPC26335-100ug Biomatik Corporation 100ug 1463 EUR

Recombinant Rabbit Tissue factor pathway inhibitor (TFPI)

RPC26335-20ug Biomatik Corporation 20ug 580.8 EUR

Tissue factor Recombinant Rabbit mAb (S-893-34)

S0B0577 Starter Biotechnology Co Ltd 10 μL Ask for price
Description: Host :Rabbit

Tissue Factor Pathway Inhibitor Recombinant Rabbit mAb

BS46527 Bioworld Biotech 50 ul 398 EUR
Description: Store at -20°C. Supplied in 50mM Tris-Glycine(pH 7.4), 0.15M NaCl, 40%Glycerol, 0.01% sodium azide and 0.05% BSA. Stable for 12 months from date of receipt.

Tissue Factor Pathway Inhibitor Recombinant Rabbit mAb

BS46979 Bioworld Biotech 50 ul 398 EUR
Description: Store at -20°C. Supplied in 50mM Tris-Glycine(pH 7.4), 0.15M NaCl, 40%Glycerol, 0.01% sodium azide and 0.05% BSA. Stable for 12 months from date of receipt.

Tissue Factor Protein, Rabbit, Recombinant (ECD, His Tag)

MBS8123288-002mg MyBiosource 0.02mg 235 EUR

Tissue Factor Protein, Rabbit, Recombinant (ECD, His Tag)

MBS8123288-5x002mg MyBiosource 5x0.02mg 915 EUR

Recombinant Rabbit Tissue factor pathway inhibitor (TFPI) (Active)

CSB-MP023437RB Cusabio 9137 mg Ask for price

Recombinant Rabbit Tissue factor pathway inhibitor (TFPI) (Active)

CSB-MP023437RB-20ug Cusabio 20ug Ask for price
Description: 25-300aa

Recombinant Rabbit Tissue factor pathway inhibitor (TFPI) (Active)

RPC26427-100ug Biomatik Corporation 100ug 543.9 EUR

Recombinant Rabbit Tissue factor pathway inhibitor (TFPI) (Active)

RPC26427-20ug Biomatik Corporation 20ug 381.6 EUR

OPCA00238-1MG - Recombinant Rabbit Tissue factor pathway inhibitor

OPCA00238-1MG Aviva Systems Biology 1mg 1977 EUR

OPCA00238-100UG - Recombinant Rabbit Tissue factor pathway inhibitor

OPCA00238-100UG Aviva Systems Biology 100ug 586 EUR

OPCA00238-20UG - Recombinant Rabbit Tissue factor pathway inhibitor

OPCA00238-20UG Aviva Systems Biology 20ug 400 EUR

Recombinant Rabbit Tissue factor pathway inhibitor Protein, His, E.coli-10ug

QP6775-ec-10ug EnQuireBio 10ug 391.2 EUR

Recombinant Rabbit Tissue factor pathway inhibitor Protein, His, E.coli-1mg

QP6775-ec-1mg EnQuireBio 1mg 2763.6 EUR

Recombinant Rabbit Tissue factor pathway inhibitor Protein, His, E.coli-50ug

QP6775-ec-50ug EnQuireBio 50ug 522 EUR

Recombinant Rabbit Tissue factor pathway inhibitor Protein, His, Yeast-1mg

QP6775-ye-1mg EnQuireBio 1mg 3296.4 EUR

Recombinant Rabbit Tissue factor pathway inhibitor Protein, His, E.coli-100ug

QP6775-ec-100ug EnQuireBio 100ug 848.4 EUR

Recombinant Rabbit Tissue factor pathway inhibitor Protein, His, E.coli-200ug

QP6775-ec-200ug EnQuireBio 200ug 1338 EUR

Recombinant Rabbit Tissue factor pathway inhibitor Protein, His, E.coli-500ug

QP6775-ec-500ug EnQuireBio 500ug 1816.8 EUR

Recombinant Rabbit Tissue factor pathway inhibitor Protein, His, Yeast-100ug

QP6775-ye-100ug EnQuireBio 100ug 945.6 EUR

Recombinant Rabbit Tissue factor pathway inhibitor Protein, His, Yeast-10ug

QP6775-ye-10ug EnQuireBio 10ug 434.4 EUR

Recombinant Rabbit Tissue factor pathway inhibitor Protein, His, Yeast-200ug

QP6775-ye-200ug EnQuireBio 200ug 1512 EUR

Recombinant Rabbit Tissue factor pathway inhibitor Protein, His, Yeast-500ug

QP6775-ye-500ug EnQuireBio 500ug 2164.8 EUR

Recombinant Rabbit Tissue factor pathway inhibitor Protein, His, Yeast-50ug

QP6775-ye-50ug EnQuireBio 50ug 576 EUR

Recombinant Tissue Factor (TF)

MBS2029924-001mg MyBiosource 0.01mg 175 EUR

Recombinant Tissue Factor (TF)

MBS2029924-005mg MyBiosource 0.05mg 310 EUR

Recombinant Tissue Factor (TF)

MBS2029924-01mg MyBiosource 0.1mg 470 EUR

Recombinant Tissue Factor (TF)

MBS2029924-02mg MyBiosource 0.2mg 575 EUR

Recombinant Tissue Factor (TF)

MBS2029924-05mg MyBiosource 0.5mg 1090 EUR

Recombinant Tissue Factor (TF)

MBS2012021-001mg MyBiosource 0.01mg 175 EUR

Recombinant Tissue Factor (TF)

MBS2012021-005mg MyBiosource 0.05mg 315 EUR

Recombinant Tissue Factor (TF)

MBS2012021-01mg MyBiosource 0.1mg 480 EUR

Recombinant Tissue Factor (TF)

MBS2012021-02mg MyBiosource 0.2mg 585 EUR

Recombinant Tissue Factor (TF)

MBS2012021-05mg MyBiosource 0.5mg 1110 EUR

Recombinant Tissue Factor (TF)

MBS2010710-001mg MyBiosource 0.01mg 175 EUR

Recombinant Tissue Factor (TF)

MBS2010710-005mg MyBiosource 0.05mg 310 EUR

Recombinant Tissue Factor (TF)

MBS2010710-01mg MyBiosource 0.1mg 470 EUR

Recombinant Tissue Factor (TF)

MBS2010710-02mg MyBiosource 0.2mg 575 EUR

Recombinant Tissue Factor (TF)

MBS2010710-05mg MyBiosource 0.5mg 1090 EUR

Recombinant Tissue Factor (TF)

MBS2010916-001mg MyBiosource 0.01mg 160 EUR

Recombinant Tissue Factor (TF)

MBS2010916-005mg MyBiosource 0.05mg 280 EUR

Recombinant Tissue Factor (TF)

MBS2010916-01mg MyBiosource 0.1mg 405 EUR

Recombinant Tissue Factor (TF)

MBS2010916-02mg MyBiosource 0.2mg 490 EUR

Recombinant Tissue Factor (TF)

MBS2010916-05mg MyBiosource 0.5mg 930 EUR

Recombinant Tissue Factor (TF)

MBS2011301-001mg MyBiosource 0.01mg 170 EUR

Recombinant Tissue Factor (TF)

MBS2011301-005mg MyBiosource 0.05mg 295 EUR

Recombinant Tissue Factor (TF)

MBS2011301-01mg MyBiosource 0.1mg 445 EUR

Recombinant Tissue Factor (TF)

MBS2011301-02mg MyBiosource 0.2mg 540 EUR

Recombinant Tissue Factor (TF)

MBS2011301-05mg MyBiosource 0.5mg 1025 EUR

Recombinant Tissue Factor (TF)

RPA524Bo01 Cloud-Clone 10ug 180 EUR

Recombinant Tissue Factor (TF)

4-RPA524Bo01 Cloud-Clone
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Description: Recombinant Bovine Tissue Factor expressed in: E.coli

Recombinant Tissue Factor (TF)

RPA524Hu01 Cloud-Clone 10ug 180 EUR

Recombinant Tissue Factor (TF)

4-RPA524Hu01 Cloud-Clone
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Description: Recombinant Human Tissue Factor expressed in: E.coli

Recombinant Tissue Factor (TF)

RPA524Mu01 Cloud-Clone 10ug 168 EUR

Recombinant Tissue Factor (TF)

4-RPA524Mu01 Cloud-Clone
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Description: Recombinant Mouse Tissue Factor expressed in: E.coli

Recombinant Tissue Factor (TF)

RPA524Po01 Cloud-Clone 10ug 164 EUR

Recombinant Tissue Factor (TF)

RPA524Ra01 Cloud-Clone 10ug 184 EUR

Recombinant Tissue Factor (TF)

4-RPA524Ra01 Cloud-Clone
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Description: Recombinant Rat Tissue Factor expressed in: E.coli

Recombinant Tissue Factor (TF)

RPA524Rb01 Cloud-Clone 10ug 152 EUR

Recombinant Tissue Factor (TF)

4-RPA524Rb01 Cloud-Clone
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Description: Recombinant Rabbit Tissue Factor expressed in: E.coli

Recombinant Tissue Factor (TF)

RPU53495-100ug Biomatik Corporation 100ug 554.4 EUR

Recombinant Tissue Factor (TF)

RPU53495-1mg Biomatik Corporation 1mg 2457 EUR

Recombinant Tissue Factor (TF)

RPU53495-50ug Biomatik Corporation 50ug 445.5 EUR

Recombinant Tissue Factor (TF)

RPU58458-100ug Biomatik Corporation 100ug 551.1 EUR

Recombinant Tissue Factor (TF)

RPU58458-1mg Biomatik Corporation 1mg 2558.4 EUR

Recombinant Tissue Factor (TF)

RPU58458-50ug Biomatik Corporation 50ug 428.5 EUR

Recombinant Tissue Factor (TF)

RPU58988-100ug Biomatik Corporation 100ug 947.4 EUR

Recombinant Tissue Factor (TF)

RPU58988-1mg Biomatik Corporation 1mg 3731.5 EUR

Recombinant Tissue Factor (TF)

RPU58988-50ug Biomatik Corporation 50ug 592 EUR

Recombinant Tissue Factor (TF)

RPU44024-100ug Biomatik Corporation 100ug 554.4 EUR

Recombinant Tissue Factor (TF)

RPU44024-1mg Biomatik Corporation 1mg 2457 EUR

Recombinant Tissue Factor (TF)

RPU44024-50ug Biomatik Corporation 50ug 445.5 EUR

Recombinant Tissue Factor (TF)

RPU44025-100ug Biomatik Corporation 100ug 517 EUR

Recombinant Tissue Factor (TF)

RPU44025-1mg Biomatik Corporation 1mg 2293.2 EUR

Recombinant Tissue Factor (TF)

RPU44025-50ug Biomatik Corporation 50ug 415.8 EUR

Recombinant Tissue Factor (TF)

RPU44026-100ug Biomatik Corporation 100ug 566.5 EUR

Recombinant Tissue Factor (TF)

RPU44026-1mg Biomatik Corporation 1mg 2511.6 EUR

Recombinant Tissue Factor (TF)

RPU44026-50ug Biomatik Corporation 50ug 455.4 EUR

Recombinant Tissue Factor (TF)

RPU44027-100ug Biomatik Corporation 100ug 468.6 EUR

Recombinant Tissue Factor (TF)

RPU44027-1mg Biomatik Corporation 1mg 2074.8 EUR

Recombinant Tissue Factor (TF)

RPU44027-50ug Biomatik Corporation 50ug 376.2 EUR

Tissue Factor Rabbit mAb

A4395-100ul Abclonal 100 ul 492 EUR

Tissue Factor Rabbit mAb

A4395-200ul Abclonal 200 ul 685.2 EUR

Tissue Factor Rabbit mAb

A4395-20ul Abclonal 20 ul 265.2 EUR

Tissue Factor Rabbit mAb

A4395-50ul Abclonal 50 ul 344.4 EUR

Tissue Factor Rabbit mAb

52668 SAB 100ul 499 EUR

Tissue Factor Rabbit mAb

59064 SAB 100ul 339 EUR

Tissue Factor Rabbit pAb

E2381361 EnoGene 100ul 225 EUR
Description: Available in various conjugation types.

Tissue Factor Rabbit mAb

E2R26161 EnoGene 100ul 255 EUR
Description: Available in various conjugation types.

Tissue Factor Rabbit mAb

E2R27360 EnoGene 100ul 255 EUR
Description: Available in various conjugation types.

Tissue Factor Rabbit mAb

E2R27361 EnoGene 100ul 255 EUR
Description: Available in various conjugation types.

Tissue Factor Rabbit mAb

E2R381361 EnoGene 100ul 275 EUR
Description: Biotin-Conjugated, FITC-Conjugated , AF350 Conjugated , AF405M-Conjugated ,AF488-Conjugated, AF514-Conjugated ,AF532-Conjugated, AF555-Conjugated ,AF568-Conjugated , HRP-Conjugated, AF405S-Conjugated, AF405L-Conjugated , AF546-Conjugated, AF594-Conjugated , AF610-Conjugated, AF635-Conjugated , AF647-Conjugated , AF680-Conjugated , AF700-Conjugated , AF750-Conjugated , AF790-Conjugated , APC-Conjugated , PE-Conjugated , Cy3-Conjugated , Cy5-Conjugated , Cy5.5-Conjugated , Cy7-Conjugated Antibody

Tissue factor Rabbit pAb

E47R4690 EnoGene 100ul 295 EUR

Tissue Factor Rabbit mAb

MBS4754094-01mL MyBiosource 0.1mL 450 EUR

Tissue Factor Rabbit mAb

MBS4754094-5x01mL MyBiosource 5x0.1mL 1540 EUR

Tissue Factor Rabbit mAb

MBS4754219-01mL MyBiosource 0.1mL 450 EUR

Tissue Factor Rabbit mAb

MBS4754219-5x01mL MyBiosource 5x0.1mL 1540 EUR

Tissue Factor Rabbit mAb

MBS4754220-01mL MyBiosource 0.1mL 450 EUR

Tissue Factor Rabbit mAb

MBS4754220-5x01mL MyBiosource 5x0.1mL 1540 EUR

Tissue Factor Rabbit mAb

MBS9467381-005mL MyBiosource 0.05mL 290 EUR

Tissue Factor Rabbit mAb

MBS9467381-01mL MyBiosource 0.1mL 435 EUR

Tissue Factor Rabbit mAb

MBS9467381-5x01mL MyBiosource 5x0.1mL 1810 EUR

Tissue Factor Rabbit pAb

MBS8542825-01mL MyBiosource 0.1mL 305 EUR

Tissue Factor Rabbit pAb

MBS8542825-01mLAF405L MyBiosource 0.1mL(AF405L) 565 EUR

Tissue Factor Rabbit pAb

MBS8542825-01mLAF405S MyBiosource 0.1mL(AF405S) 565 EUR

Tissue Factor Rabbit pAb

MBS8542825-01mLAF610 MyBiosource 0.1mL(AF610) 565 EUR

Tissue Factor Rabbit pAb

MBS8542825-01mLAF635 MyBiosource 0.1mL(AF635) 565 EUR

Recombinant Human Tissue factor

MBS7609429-005mg MyBiosource 0.05mg 405 EUR

Recombinant Human Tissue factor

MBS7609429-02mg MyBiosource 0.2mg 760 EUR

Recombinant Human Tissue factor

MBS7609429-1mg MyBiosource 1mg 2175 EUR

Recombinant Human Tissue factor

MBS7609429-5x1mg MyBiosource 5x1mg 8410 EUR

Recombinant Human Tissue factor

MBS967694-005mgBaculovirus MyBiosource 0.05mg(Baculovirus) 1125 EUR

Recombinant Human Tissue factor

MBS967694-005mgEColi MyBiosource 0.05mg(E-Coli) 260 EUR

Recombinant Human Tissue factor

MBS967694-02mgEColi MyBiosource 0.2mg(E-Coli) 560 EUR

Recombinant Human Tissue factor

MBS967694-05mgEColi MyBiosource 0.5mg(E-Coli) 875 EUR

Recombinant Human Tissue factor

MBS967694-1mgEColi MyBiosource 1mg(E-Coli) 1325 EUR

Tissue Factor Recombinant Protein

40-663 ProSci 2 ug 311.1 EUR
Description: Tissue factor is a transmembrane glycoprotein of the cytokine receptor superfamily that acts as a receptor for coagulation factor VII (fVII) to trigger initiation of the coagulation cascade in response to vascular injury. Expression of tissue factor occurs constitutively within most extravascular and perivascular cells and at high levels within critical organs and tissue. Tissue factor is not normally expressed freely on the surface of circulating blood cells due to its pro-coagulant effect, but is instead stored on the surface of mononuclear and endothelial cells in microparticles that can shed into circulation in response to vascular injury, pro-inflammatory cytokines, or microbial ligands. Tissue factor can also be shed into circulation by cancer cells where its expression in a number of cancer types has been linked to tumor progression, metastatic potential, thrombosis, and angiogenesis. Expression of tissue factor has been shown to be inducible by select cytokines in a number of cell types, including IL-1β and TNF-α in vascular endothelial cells and macrophages, and TNF-α, IL-6, and FGF-Basic in monocytes, among others. CHO cell-derived Recombinant Human Tissue Factor is a glycoprotein homodimer comprised of the 214-amino-acid length monomer containing a C-terminal His-Tag. It has a calculated molecular weight of approximately 24.4 kDa, and as a result of glycosylation, Recombinant Human Tissue Factor migrates with an apparent molecular mass of approximately 45-55 kDa by SDS-PAGE gel, under reducing conditions.

Rabbit tissue factor X ELISA

E01A34388 BlueGene 96T 700 EUR
Description: ELISA

Rabbit tissue factor X ELISA

E04T0135-48wellsplate BlueGene 48 wells plate 280 EUR

Rabbit tissue factor X ELISA

E04T0135-96wellsplate BlueGene 96 wells plate 405 EUR

Rabbit Tissue Factor ELISA kit

E01A34338 BlueGene 96T 700 EUR
Description: ELISA

Rabbit tissue factor VII ELISA

E01A34385 BlueGene 96T 700 EUR
Description: ELISA

Rabbit Tissue Factor ELISA Kit

MBS034222-INQUIRE MyBiosource INQUIRE Ask for price

Rabbit Tissue factor ELISA Kit

ELA-E0524Rb Lifescience Market 96 Tests 1113.6 EUR

Rabbit tissue factor VII ELISA

E04T0131-48wellsplate BlueGene 48 wells plate 280 EUR

Rabbit tissue factor VII ELISA

E04T0131-96wellsplate BlueGene 96 wells plate 405 EUR

Rabbit Tissue Factor ELISA kit

E04T0037-192T BlueGene 192 tests 1524 EUR
Description: A competitive ELISA for quantitative measurement of Rabbit Tissue Factor in samples from blood, plasma, serum, cell culture supernatant and other biological fluids. This is a high quality ELISA kit developped for optimal performance with samples from the particular species.

Rabbit Tissue Factor ELISA kit

E04T0037-48 BlueGene 1 plate of 48 wells 624 EUR
Description: A competitive ELISA for quantitative measurement of Rabbit Tissue Factor in samples from blood, plasma, serum, cell culture supernatant and other biological fluids. This is a high quality ELISA kit developped for optimal performance with samples from the particular species.

Rabbit Tissue Factor ELISA kit

E04T0037-48wellsplate BlueGene 48 wells plate 280 EUR

Rabbit Tissue Factor ELISA kit

E04T0037-96 BlueGene 1 plate of 96 wells 822 EUR
Description: A competitive ELISA for quantitative measurement of Rabbit Tissue Factor in samples from blood, plasma, serum, cell culture supernatant and other biological fluids. This is a high quality ELISA kit developped for optimal performance with samples from the particular species.

Rabbit Tissue Factor ELISA kit

E04T0037-96wellsplate BlueGene 96 wells plate 405 EUR

Rabbit Tissue Factor ELISA Kit

MBS725252-10x96StripWells MyBiosource 10x96-Strip-Wells 5685 EUR

Rabbit Tissue Factor ELISA Kit

MBS725252-48StripWells MyBiosource 48-Strip-Wells 485 EUR
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Per ogni famiglia ci sono 3 isotipi (α, β, γ) e per ogni isotipo diverse isoforme. Ogni NRR è composto da 6 regioni (A-F). 3 regioni sono importanti: la regione A / B ha una funzione di attivazione trascrizionale indipendente dal ligando, la regione C ospita il dominio di legame del DNA, la regione E ospita il dominio di legame del ligando. Per regolare l’espressione dei geni bersaglio, NRR deve dimerizzare. RXR sono obbligatori nei dimeri (eterodimeri RAR-RXR, omodimeri RXR-RXR). I dimeri si legano a specifiche sequenze di DNA, presenti nei promotori dei geni bersaglio. Quando il ligando, naturale o sintetico, si lega all’RNR, vengono reclutati i coattivatori e vengono attivati ​​i fattori di trascrizione. Nella cellula bersaglio, i retinoidi non utilizzati vengono degradati nei metaboliti polari dagli enzimi del citocromo P450.

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